Membrane Transporter Proteins

Membrane transport proteins, also known as membrane transport proteins, selectively transport small molecules across the plasma membrane that are not freely diffusing. Membrane transport proteins are membrane integral proteins, or large transmembrane molecular complexes, that function to participate in passive or active transport.

Cat. No.	Product name
BP16101	Norverapamil hydrochloride
BP16101	Norverapamil hydrochloride ((±)-Norverapamil hydrochloride) is an N-demethylated metabolite of Verapamil and it is an L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor.
BP16102	NP118809
BP16102	NP118809 is a potent N-type calcium channel blocker(IC50 : 0.11 μM).
BP16103	NS11394
BP16103	NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(1) at GABA(A) alpha subunit-containing receptors.
BP16104	NS13001
BP16104	NS13001 is a potent, selective, orally active allosteric positive modulator of SK channels (small conductance calcium-activated potassium channels). The EC50s are 1.8 and 0.14 μM for SK2 and SK3, respectively. NS13001 holds promise as a potential therapeutic agent for treatment of spinocerebellar ataxia type 2 (SCA2) and possibly other cerebellar ataxias.
BP16105	NS1652
BP16105	NS1652 is an anion conductance inhibitor. NS1652 blocks chloride channel has an IC50 of 1.6 μM in human and mouse red blood cells.
BP16106	NS19504
BP16106	NS19504 is an activator of Ca2+-activated K+ channel with EC50 of 11.0 µM. NS19504 shows relaxing effect on bladder smooth muscle spontaneous phasic contractions.
BP16107	NS6180
BP16107	NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.
BP16108	NS8593 hydrochloride
BP16108	NS8593 hydrochloride is a potent and selective inhibitor of small conductance Ca2+-activated K+ channels (SK channels).
BP16109	Oleoyl Serotonin
BP16109	Oleoyl Serotonin is an antagonist of hTRPV1 with an IC50 of 2.57 μM.
BP16110	Oligomycin A
BP16110	Oligomycin A is an inhibitor of ATP synthase, inhibits oxidative phosphorylation and all the ATP-dependent processes occurring on the coupling membrane of mitochondria.
BP16111	Olvanil
BP16111	Olvanil is a vanilloid receptor agonist with EC50 of 0.7nM.
BP16112	Omeprazole sulfide
BP16112	Omeprazole sulfide is a metabolite of Omeprazole, which is a proton pump inhibitor.
BP16113	Oxiracetam
BP16113	Oxiracetam, a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.
BP16114	Oxybutynin chloride
BP16114	Oxybutynin is an anticholinergic medication used to relieve urinary and bladder difficulties. It competitively antagonizes the M1, M2, and M3 subtypes of the muscarinic acetylcholine receptor.
BP16115	Pagoclone
BP16115	Pagoclone is a GABA receptor agonist and can be used for studies on the treatment of stuttering, panic disorder, and generalized anxiety. Pagoclone is a partial agonist at α1-, α2- and α5-containing GABAA receptors and a full agonist at receptors containi
BP16116	PAP-1
BP16116	PAP-1 is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).
BP16117	PEAQX
BP16117	PEAQX(NVP-AAM 077) is an effective and orally available NMDA antagonist. It can inhibit human NMDA receptors for 1A/2A(IC50: 270 nM), rather than 1A/2B(29, 600 nM).
BP16118	Pepluanin A
BP16118	Pepluanin A, shows a very high activity for a jatrophane diterpene, outperforming cyclosporin A by a factor of at least 2 in the inhibition of Pgp-mediated daunomycin transport.
BP16119	Periplocymarin
BP16119	Periplocymarin, a cardiac glycoside, has potential anti-cancer activity.
BP16120	Permethrin
BP16120	Permethrin is a pyrethroid insecticide commonly used in the treatment of LICE INFESTATIONS and SCABIES.