TAS-120 is a novel, potent and highly selective FGFR inhibitor, used for antitumor treatment.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 113 | |
2 mg | In stock | $ 214 | |
4 mg | In stock | $ 307 | |
10 mg | In stock | $ 666 | |
20 mg | In stock | $ 1018 |
Description | TAS-120 is a novel, potent and highly selective FGFR inhibitor, used for antitumor treatment. |
Targets&IC50 | FGFR2 E566G: 2.4 nM (IC50), FGFR2 N550H: 3.6 nM (IC50), FGFR4: 8.3 nM (IC50), FGFR3: 1.6 nM (IC50), wild-type FGFR2: 0.3 nM (IC50), FGFR2 V5651: 1-3 nM (IC50), FGFR1: 3.9 nM (IC50), FGFR2: 1.3 nM (IC50) |
Synonyms | FGFR-IN-1, TAS120 |
CAS No. | 1448169-71-8 |
Chemical Formula | C22H22N6O3 |
Molecular Weight | 418.457 |
Solubility | DMSO: 29 mg/mL (69.30 mM) |
Storage | Powder: -20°C for 2 years In solvent: -80°C for 1 year |
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