BP13189
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DUB-IN-2
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Dub-in-2, with an IC50 value of 0.28 for USP8, is an effective deubiquitinase inhibitor.
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BP13190
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DUB-IN-3
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DUB-IN-3 is a potent deubiquitinase (USP) enzyme inhibitor extracted from reference compound 22c. The IC50 for USP8 is 0.56 μM.
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BP13191
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dUTP trisodium
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dUTP trisodium is a deoxyuridine phosphate having a triphosphate group at the 5'-position and can be used for PCR.
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BP13192
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DYRKs-IN-1
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DYRKs-IN-1 has antitumor activity. DYRKs-IN-1 is a potent DYRKs (Dual-specificity tyrosine-phosphorylation-regulated kinases) inhibitor with IC50s of 9 nM and 5 nM for DYRK1B and DYRK1A, respectively.
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BP13193
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DYRKs-IN-2
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DYRKs-IN-2 has antitumor activity. DYRKs-IN-2 is a potent DYRKs inhibitor with IC50s of 30.6 nM and 12.8 nM for DYRK1B and DYRK1A, respectively.
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BP13194
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E3330
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E3330 is a potent and selective APE1(Ref-1) inhibitor, which suppressed NF-kappa B DNA-binding activity.
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BP13195
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Eciruciclib
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Eciruciclib is an inhibitor of CDK with antitumor properties.
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BP13196
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Tomivosertib
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eFT508 is a potent, highly selective MNK1 and MNK2 inhibitor with IC50 value of 1-2 nM.
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BP13197
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EHop-016
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EHop-016 is a specific Rac GTPase inhibitor with IC50 of 1.1 μM for Rac1 in MDA-MB-231 and MDA-MB-435 cells, equally effective inhibition for Rac3.
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BP13198
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EHT 1864
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EHT 1864 is a effective Rac family GTPase inhibitor for Rac1/Rac1b/Rac2/Rac3 (Kd: 40/50/60/250 nM).
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BP13199
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EHT 1610
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EHT 5372 is a strong DYRK’s family kinases of inhibitor (IC50s: 0.22, 0.28 nM for DYRK1A and DYRK1B, respectively).
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BP13200
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EN4
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EN4 MYC inhibitor is a covalent ligand that targets cysteine 171 (C171) of MYC. It is selective for c-MYC over N-MYC and L-MYC, and inhibits MYC transcriptional activity, downregulates MYC targets, and impairs tumorigenesis.
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BP13201
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Enocitabine
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Enocitabine is a nucleoside analog. Enocitabine inhibits the replication of human cytomegalovirus(HCMV) and it also has antileukemic and antiviral activities. Enocitabine is also a potent DNA replication inhibitor and a DNA chain terminator.
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BP13202
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Enoxacin
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Enoxacin is a broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.
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BP13203
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Enoxacin hydrate
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Enoxacin is a broad-spectrum 6-fluoronaphthyridinone antibacterial agent.
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BP13204
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Enrofloxacin
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Enrofloxacin is a veterinary antibacterial agent, used in poultry.
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BP13205
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EOAI3402143
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EOAI3402143 inhibits Usp9x and Usp24 activity, increases tumor cell apoptosis. EOAI3402143 phenocopies the FAS induction and apoptotic sensitization of Usp5 knockdown and fully blocks melanoma tumor growth.
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BP13206
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Epirubicin hydrochloride
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Epirubicin hydrochloride is an antineoplastic agent which can inhibit Topoisomerase.
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BP13207
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Vitamin D2
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Ergocalciferol (Vitamin D2) is a derivative of ergosterol formed by ultraviolet rays breaking of the C9-C10 bond with a strong inhibitory effect against bladder tumor promotion by sodium saccharin, and it induces cell differentiation in leukemia cells. Vitamin D2 is an inhibitor of DNA Polymerase.
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BP13208
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Ethynylcytidine
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Ethynylcytidine is a nucleoside antimetabolite.
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