BP13589
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Y16
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Y16 is a G-protein–coupled Rho GEFs inhibitor; works synergistically with Rhosin/G04 in inhibiting LARG-RhoA interaction, RhoA activation, and RhoA-mediated signaling functions.
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BP13590
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Y16 acetate(429653-73-6 free base)
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Y16 is a G-protein–coupled Rho GEFs inhibitor; works synergistically with Rhosin/G04 in inhibiting LARG-RhoA interaction, RhoA activation, and RhoA-mediated signaling functions.
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BP13591
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Y-33075 dihydrochloride
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Y-33075 dihydrochloride is a selective inhibitor of ROCK(IC50 of 3.6 nM).
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BP13592
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YKL-5-124
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YKL-5-124, a potent, selective and covalent CDK7 inhibitor with an IC50 of 9.7 nM, 1300 nM and 3020 nM for CDK7/Mat1/CycH, CDK2 and CDK9 respectively, displays biochemical and cellular selectivity for CDK7 over CDK12/13.
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BP13593
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YM-46303
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YM-46303 is an antagonist of mAChR
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BP13594
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ZCL278
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ZCL278 is a selective Cdc42 GTPase inhibitor.
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BP13595
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ZD 7155(hydrochloride)
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ZD 7155 hydrochloride is an antagonist of angiotensin II receptor type 1 (AT1 receptor).
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BP13596
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ZINC00881524
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ZINC00881524 is an effective and specific ROCK inhibitor.
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BP13597
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ZINC69391
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ZINC69391 is a selective inhibitor of Rac1 with antiproliferative and antimetastatic effects. ZINC69391 interferes with the interaction of Rac1 with Dock180, reduces Rac1-GTP levels and induces apoptosis.
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BP13598
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ZN-c3
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ZN-c3 is a potent and selective Wee1 inhibitor with balanced potency, ADME, and pharmacokinetic properties.
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BP13599
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Zoliflodacin
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Zoliflodacin (ETX0914, AZD0914) is a new bacterial DNA gyrase/topoisomerase inhibitor. Zoliflodacin has potent in vitro antibacterial activity against Gram-positive and Gram-negative organisms, including S. aureus (MIC90: 0.25 μg/mL).
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BP13600
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ZYN57939
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ZYN57939 is RNA polymerase I inhibitor for treating RNA polymerase I- mediated diseases. ZYN57939 showed inhibitory activity with IC50 of 0.855 μM against human HT- 29 cancer cell lines.
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BP13601
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H-1152 dihydrochloride
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