GSK9311 hydrochloride, a less active analog of GSK6853, can be used as a negative control. GSK9311 hydrochloride inhibits BRPF bromodomain (pIC50s: 6.0 and 4.3 for BRPF1 and BRPF2).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | 6-8 weeks | $ 1015 | |
10 mg | 6-8 weeks | $ 1928 | |
20 mg | 6-8 weeks | $ 2892 | |
50 mg | 6-8 weeks | $ 5697 | |
100 mg | 6-8 weeks | $ 8830 |
Description | GSK9311 hydrochloride, a less active analog of GSK6853, can be used as a negative control. GSK9311 hydrochloride inhibits BRPF bromodomain (pIC50s: 6.0 and 4.3 for BRPF1 and BRPF2). |
Targets&IC50 | BRPF2:4.3(pIC50), BRPF1:6(pIC50) |
In vitro | GSK6853 is a less active analogue of GSK6853 in which the 5-amide is alkylated.GSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain, and demonstrates properties suitable for cellular and in vivo studies. |
CAS No. | 2253733-09-2 |
Chemical Formula | C24H32ClN5O3 |
Molecular Weight | 474 |
Storage | Powder: -20°C for 2 years In solvent: -80°C for 1 year |
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