Aurora kinase inhibitor III is a potent inhibitor of Aurora A kinase (IC50 = 42 nM).1 It is selective for Aurora A over BMX, BTK, IGF-1R, c-Src, TRKB, SYK, and EGFR.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 134 | |
2 mg | In stock | $ 241 | |
4 mg | In stock | $ 385 | |
10 mg | In stock | $ 754 | |
20 mg | In stock | $ 1138 |
Description | Aurora kinase inhibitor III is a potent inhibitor of Aurora A kinase (IC50 = 42 nM).1 It is selective for Aurora A over BMX, BTK, IGF-1R, c-Src, TRKB, SYK, and EGFR. |
Targets&IC50 | Aurora A:42 nM |
Synonyms | Aurora Kinase Inhibitor III |
CAS No. | 879127-16-9 |
Chemical Formula | C21H18F3N5O |
Molecular Weight | 413.404 |
Solubility | DMSO: 50 mg/mL (120.9 mM) |
Storage | Powder: -20°C for 2 years In solvent: -80°C for 1 year |
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