CaMKII-IN-1 is a potent and highly selective inhibitor of CaMKII (IC50 = 63 nM). CaMKII-IN-1 exhibited more than 100-fold higher selectivity for CaMKII over CaMKIV, MLCK, p38a, Akt1, and PKC.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | In stock | $ 293 | |
4 mg | In stock | $ 527 | |
8 mg | In stock | $ 778 | |
20 mg | In stock | $ 1697 | |
40 mg | In stock | $ 2681 |
Description | CaMKII-IN-1 is a potent and highly selective inhibitor of CaMKII (IC50 = 63 nM). CaMKII-IN-1 exhibited more than 100-fold higher selectivity for CaMKII over CaMKIV, MLCK, p38a, Akt1, and PKC. |
Targets&IC50 | CaMKII:63 nM |
CAS No. | 1208123-85-6 |
Chemical Formula | C29H30ClN5O2S |
Molecular Weight | 548.1 |
Solubility | DMSO: 54 mg/mL (98.52 mM) |
Storage | Powder: -20°C for 2 years In solvent: -80°C for 1 year |
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