K-252c is a staurosporine analog isolated from Nocardiopsis sp. and is a cell-permeable PKC inhibitor (IC50: 2.45 μM). K-252c also inhibits β-lactamase, chymotrypsin, and malate dehydrogenase. K-252c causes apoptosis in human chronic myelogenous leukemia cancer cells.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | 2-3 weeks | $ 1177 | |
10 mg | 2-3 weeks | $ 2236 | |
20 mg | 2-3 weeks | $ 3577 | |
50 mg | 2-3 weeks | $ 6226 | |
100 mg | 2-3 weeks | $ 9401 |
Description | K-252c is a staurosporine analog isolated from Nocardiopsis sp. and is a cell-permeable PKC inhibitor (IC50: 2.45 μM). K-252c also inhibits β-lactamase, chymotrypsin, and malate dehydrogenase. K-252c causes apoptosis in human chronic myelogenous leukemia cancer cells. |
Targets&IC50 | PKC:2.45 μM |
CAS No. | 85753-43-1 |
Chemical Formula | C20H13N3O |
Molecular Weight | 311.344 |
Storage | Powder: -20°C for 2 years In solvent: -80°C for 1 year |
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